Triazole-based estradiol dimers prepared via CuAAC from 17α-ethinyl estradiol with five-atom linkers causing G2/M arrest and tubulin inhibition-Reference-Cited by-同舟云学术

Triazole-based estradiol dimers prepared via CuAAC from 17α-ethinyl estradiol with five-atom linkers causing G2/M arrest and tubulin inhibition

Published:2023-02 Issue: Volume:131 Page:106334
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Jurášek Michal,Řehulka Jiří,Hrubá Lenka,Ivanová Aleksandra,Gurská Soňa,Mokshyna Olena,Trousil Pavel,Huml Lukáš,Polishchuk Pavel,Hajdúch Marián,Drašar Pavel B.,Džubák Petr

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference31 articles.

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2. Polymer-free corticosteroid dimer implants for controlled and sustained drug delivery;Battiston;Nat. Commun.,2021

3. Radioiodinated estradiol dimer for estrogen receptor targeted breast cancer imaging;Xu;Chem. Biol. Drug. Des.,2020

4. A review on steroid dimers: 2011–2019;Nahar;Steroids,2020

5. Estradiol dimer inhibits tubulin polymerization and microtubule dynamics;Jurášek;J. Steroid. Biochem. Mol. Biol.,2018

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