Synthesis and biological evaluation of thieno[3,2-c]pyrazol-3-amine derivatives as potent glycogen synthase kinase 3β inhibitors for Alzheimer’s disease-Reference-Cited by-同舟云学术

Synthesis and biological evaluation of thieno[3,2-c]pyrazol-3-amine derivatives as potent glycogen synthase kinase 3β inhibitors for Alzheimer’s disease

Published:2023-09 Issue: Volume:138 Page:106663
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Yan Ning,Xie Fei,Tang Long-Qian,Wang De-Feng,Li Xiang,Liu Chao^ORCID,Liu Zhao-Peng

Funder

Key Technology Research and Development Program of Shandong Province

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference79 articles.

1. C. Patterson, World Alzheimer Report 2018. London: Alzheimer's Disease International, 2018. https://www.alzint.org/resource/world-alzheimer-report-2018.

2. S. Gauthier, P. Rosa-Neto, J.A. Morais, C. Webster, World Alzheimer Report 2021. London: Alzheimer's Disease International, 2021. https://www.alzint.org/resource/world-alzheimer-report-2021.

3. Recent advances on drug development and emerging therapeutic agents for Alzheimer's disease;Athar;Mol. Biol. Rep.,2021

4. Sodium oligomannate: first approval;Syed;Drugs,2020

5. Aducanumab: first approval;Dhillon;Drugs,2021

Cited by 6 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design, synthesis and biological evaluation of thieno[3,2-c]pyrazol-urea derivatives as potent glycogen synthase kinase 3β inhibitors based on the DFG-out conformation;Bioorganic & Medicinal Chemistry Letters;2024-11

2. New insights into butyrylcholinesterase: Pharmaceutical applications, selective inhibitors and multitarget-directed ligands;European Journal of Medicinal Chemistry;2024-09

3. Identification of vilazodone as a novel plasminogen activator inhibitor to overcome Alzheimer's disease through virtual screening, molecular dynamics simulation, and biological evaluation;Archiv der Pharmazie;2024-05-30

4. The classical D1 dopamine receptor antagonist SCH23390 is a functional sigma-1 receptor allosteric modulator;Acta Pharmacologica Sinica;2024-04-11

5. Fused thiophene as a privileged scaffold: A review on anti-Alzheimer's disease potentials via targeting cholinesterases, monoamine oxidases, glycogen synthase kinase-3, and Aβ aggregation;International Journal of Biological Macromolecules;2024-04