Unique binding pocket for KW-4679 in the histamine H1 receptor
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference28 articles.
1. Heterogeneity of the M1 muscarinic receptor subtype between peripheral lung and cerebral cortex demonstrated by the selective antagonist AF-DX 116;Bloom;Life Sci.,1987
2. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50% inhibition (IC50) of an enzymatic reaction;Cheng;Biochem. Pharmacol.,1973
3. Binding of antidepressants to human brain receptors: focus on newer generation compounds;Cusack;Psychopharmacology,1994
4. In vitro and in vivo studies of the non-sedating antihistamine epinastine;Fügner;Arzneim.-Forsch. Drug Res.,1988
5. Specific binding of [3H]-thiotidine to histamine H2 receptors in guinea pig cerebral cortex;Gajtkowski;Nature,1983
Cited by 63 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Pharmacological Characterization of the Zebrafish (Danio Rerio) Histamine H1Receptor Reveals the Involvement of the Second Extracellular Loop in the Binding of Histamine;Molecular Pharmacology;2023-11-17
2. Etiology and pharmacotherapy of ocular surface allergic diseases;Handbook of Basic and Clinical Ocular Pharmacology and Therapeutics;2022
3. Discovery to Launch of Anti-allergy (Emadine; Patanol/Pataday/Pazeo) and Anti-glaucoma (Travatan; Simbrinza) Ocular Drugs, and Generation of Novel Pharmacological Tools Such as AL-8810;ACS Pharmacology & Translational Science;2020-11-05
4. Roles of Lys191 and Lys179 in regulating thermodynamic binding forces of ligands to determine their binding affinity for human histamine H1 receptors;Biochemical Pharmacology;2020-10
5. Asymmetric Catalysis upon Helically Chiral Loratadine Analogues Unveils Enantiomer-Dependent Antihistamine Activity;Journal of the American Chemical Society;2020-06-24
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3