Novel, highly potent PROTACs targeting AURORA-A kinase-Reference-Cited by-同舟云学术

Novel, highly potent PROTACs targeting AURORA-A kinase

Published:2022 Issue: Volume:2 Page:100032
ISSN:2666-2469
Container-title:Current Research in Chemical Biology
language:en
Short-container-title:Current Research in Chemical Biology

Author:

Bozilovic Jelena,Eing Lorenz,Berger Benedict-Tilman,Adhikari Bikash,Weckesser Janik,Berner Nicola B.,Wilhelm Stephanie,Kuster Bernhard,Wolf Elmar,Knapp Stefan^ORCID

Publisher

Elsevier BV

Subject

General Engineering

Reference42 articles.

1. PROTAC-mediated degradation reveals a non-catalytic function of AURORA-A kinase;Adhikari;Nat. Chem. Biol.,2020

2. A phase I study of MK-5108, an oral aurora a kinase inhibitor, administered both as monotherapy and in combination with docetaxel, in patients with advanced or refractory solid tumors;Amin;Invest. N. Drugs,2016

3. PROTAC targeted protein degraders: the past is prologue;Bekes;Nat. Rev. Drug Discov.,2022

4. A phase II trial of the aurora kinase A inhibitor alisertib for patients with castration-resistant and neuroendocrine prostate cancer: efficacy and biomarkers;Beltran;Clin. Cancer Res.,2019

5. Robust, reproducible and quantitative analysis of thousands of proteomes by micro-flow LC-MS/MS;Bian;Nature Communications,2020

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3. Metabolic protein kinase signalling in neuroblastoma;Molecular Metabolism;2023-09

4. Targeted protein degradation in cancers: Orthodox PROTACs and beyond;The Innovation;2023-05

5. Targeted AURKA degradation: Towards new therapeutic agents for neuroblastoma;European Journal of Medicinal Chemistry;2023-02