Impact of Extensive Plasma Protein Binding on the In Situ Hepatic Uptake and Clearance of Perampanel and Fluoxetine in Sprague Dawley Rats-Reference-Cited by-同舟云学术

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Impact of Extensive Plasma Protein Binding on the In Situ Hepatic Uptake and Clearance of Perampanel and Fluoxetine in Sprague Dawley Rats

Published:2020-10 Issue:10 Volume:109 Page:3190-3205
ISSN:0022-3549
Container-title:Journal of Pharmaceutical Sciences
language:en
Short-container-title:Journal of Pharmaceutical Sciences

Author:

Bteich Michel,Poulin Patrick,Piette Sarah,Haddad Sami

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference75 articles.

1. Transporter-induced protein binding shift (TIPBS) hypothesis and modeling;Baik,2015

2. Plasma/serum protein binding determinations;Banker;Curr Drug Metabol,2008

3. Protein binding in plasma: a case history of a highly protein-bound drug;Barnaby,2004

4. BDDCS applied to over 900 drugs;Benet;AAPS J,2011

5. The isolated perfused rat liver: standardization of a time-honoured model;Bessems;Lab Anim,2006

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Plasma protein-mediated uptake and contradictions to the free drug hypothesis: a critical review;Drug Metabolism Reviews;2023-04-12

2. The structural basis for high affinity binding of α1-acid glycoprotein to the potent antitumor compound UCN-01;Journal of Biological Chemistry;2021-12

3. A New Guidance for the Prediction of Hepatic Clearance in the Early Drug Discovery and Development from the in Vitro-to-in Vivo Extrapolation Method and an Approach for Exploring Whether an Albumin-Mediated Hepatic Uptake Phenomenon Could be Present Under in Vivo Conditions;Journal of Pharmaceutical Sciences;2021-07

4. Comparative Assessment of Extrapolation Methods Based on the Conventional Free Drug Hypothesis and Plasma Protein-Mediated Hepatic Uptake Theory for the Hepatic Clearance Predictions of Two Drugs Extensively Bound to Both the Albumin And Alpha-1-Acid Glycoprotein;Journal of Pharmaceutical Sciences;2021-03

5. Albumin-Mediated Uptake Improves Human Clearance Prediction for Hepatic Uptake Transporter Substrates Aiding a Mechanistic In Vitro-In Vivo Extrapolation (IVIVE) Strategy in Discovery Research;The AAPS Journal;2020-11-16

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