The importance of target binding kinetics for measuring target binding affinity in drug discovery: a case study from a CRF1 receptor antagonist program-Reference-Cited by-同舟云学术

The importance of target binding kinetics for measuring target binding affinity in drug discovery: a case study from a CRF1 receptor antagonist program

Published:2020-01 Issue:1 Volume:25 Page:7-14
ISSN:1359-6446
Container-title:Drug Discovery Today
language:en
Short-container-title:Drug Discovery Today

Author:

Hoare Sam R.J.,Fleck Beth A.^ORCID,Williams John P.,Grigoriadis Dimitri E.

Publisher

Elsevier BV

Subject

Drug Discovery,Pharmacology

Reference53 articles.

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4. Binding kinetics and mechanism of action: toward the discovery and development of better and best in class drugs;Zhang;Expert Opin. Drug Discov.,2010

5. Drug–target kinetics in drug discovery;Tonge;ACS Chem. Neurosci.,2018

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