Strategy for the Thermostabilization of an Agonist-Bound GPCR Coupled to a G Protein-Reference-Cited by-同舟云学术

Strategy for the Thermostabilization of an Agonist-Bound GPCR Coupled to a G Protein

Published:2017 Issue: Volume: Page:243-264
ISSN:0076-6879
Container-title:Methods in Enzymology
language:
Short-container-title:

Author:

Strege Annette,Carpenter Byron,Edwards Patricia C.,Tate Christopher G.

Publisher

Elsevier

Reference38 articles.

1. Structure of the adenosine A(2A) receptor bound to an engineered G protein;Carpenter;Nature,2016

2. Engineering a minimal G protein to facilitate crystallisation of G protein-coupled receptors in their active conformation;Carpenter;Protein Engineering, Design & Selection,2016

3. Progress in structure based drug design for G protein-coupled receptors;Congreve;Journal of Medicinal Chemistry,2011

4. Structure of class C GPCR metabotropic glutamate receptor 5 transmembrane domain;Dore;Nature,2014

5. Structure of the adenosine A(2A) receptor in complex with ZM241385 and the xanthines XAC and caffeine;Dore;Structure,2011

Cited by 11 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Finding the Perfect Fit: Conformational Biosensors to Determine the Efficacy of GPCR Ligands;ACS Pharmacology & Translational Science;2022-08-14

2. Structure and activity of a thermally stable mutant of Acanthamoeba actophorin;Acta Crystallographica Section F Structural Biology Communications;2022-03-28

3. ThermoFRET: A novel nanoscale G protein coupled receptor thermostability assay functional in crude solubilised membrane preparations;2020-07-08

4. Cryo-Electron Microscopy: Moving Beyond X-Ray Crystal Structures for Drug Receptors and Drug Development;Annual Review of Pharmacology and Toxicology;2020-01-06

5. Cryo-EM structures of GPCRs coupled to Gs, Gi and Go;Molecular and Cellular Endocrinology;2019-05