Highly regioselective synthesis of 2,3-disubstituted 2 H -1-benzopyrans: Brønsted acid catalyzed [4+2] cycloaddition reaction with a variety of arylalkynes via ortho -quinone methides-Reference-Cited by-同舟云学术

Highly regioselective synthesis of 2,3-disubstituted 2 H -1-benzopyrans: Brønsted acid catalyzed [4+2] cycloaddition reaction with a variety of arylalkynes via ortho -quinone methides

Published:2017-11 Issue:45 Volume:73 Page:6456-6464
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Tanaka Kenta,Sukekawa Mayumi,Shigematsu Yosuke,Hoshino Yujiro,Honda Kiyoshi

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference49 articles.

1. Structure-activity relationship of antiestrogens. Studies on 2,3-diaryl-1-benzopyrans

2. Structure-activity relationship of antiestrogens. Effect of the side chain and its position on activity of 2,3-diaryl-2H-1-benzopyrans

3. Structure-activity relationship of antiestrogens. Phenolic analogs of 2,3-diaryl-2H-1-benzopyrans

4. Synthesis and structure–activity relationships of analogs of EM-652 (acolbifene), a pure selective estrogen receptor modulator. Study of nitrogen substitution

5. (S)-(+)-4-[7-(2,2-Dimethyl-1-oxopro- poxy)-4-methyl-2-[4-[2-(1-piperidinyl)- ethoxy]phenyl]-2H-1-benzopyran-3-yl]- phenyl 2,2-Dimethylpropanoate (EM-800): A Highly Potent, Specific, and Orally Active Nonsteroidal Antiestrogen

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