1. Proteinase Inhibitors;Powers,1986
2. Diphenyl 1-Aminoalkanephosphonates
3. Abbreviations: Ac, acetyl; Boc, tert-butyloxycarbonyl; Cat G, cathepsin G; Cbz, benzyloxycarbonyl; CDI, carbonyldiimidazole; DCC, dicyclohexylcarbodiimide; DCU, dicyclohexylurea; DFP, diisopropyl ftuorophosphate; Dpa, β,β-diphenylphenylalanine; DPP-IV, dipeptidyl-peptidase IV; Et, ethyl; HEPES, 4-(2-hydroxyethyl)1-piperazineethanesulfonic acid; HLE, human leukocyte elastase; Me, methyl; pNA, p-nitroanilide; Nva, norvaline; Ph, phenyl; PhGly, phenylglycine; RMCP II, rat mast cell protease II; Suc, succinyl; TLC, thin-layer chromatography.
4. Irreversible inhibition of serine proteases by peptide derivatives of (.alpha.-aminoalkyl)phosphonate diphenyl esters
5. Synthesis of phosphonopeptides as thrombin inhibitors