Dynamics of ligand binding to GPCR: Residence time of melanocortins and its modulation
Author:
Funder
Estonian Ministry of Education and Science
European Union
Publisher
Elsevier BV
Subject
Pharmacology
Reference47 articles.
1. The druggable genome: evaluation of drug targets in clinical trials suggests major shifts in molecular class and indication;Rask-Andersen;Annu. Rev. Pharmacol. Toxicol.,2014
2. Drug-target residence time and its implications for lead optimization;Copeland;Nat. Rev. Drug Discov.,2006
3. The uptake of atropine and related drugs by intestinal smooth muscle of the guinea-pig in relation to acetylcholine receptors;Paton;Proc. R. Soc. Lond. [Biol.],1965
4. Drug-target residence time – a case for G protein-coupled receptors;Guo;Med. Res. Rev.,2014
5. Scintillation proximity assay: a sensitive and continuous isotopic method for monitoring ligand/receptor and antigen/antibody interactions;Udenfriend;Anal. Biochem.,1987
Cited by 8 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3;Journal of Medicinal Chemistry;2023-10-31
2. Ligand-Free Signaling of G-Protein-Coupled Receptors: Physiology, Pharmacology, and Genetics;Molecules;2023-08-31
3. Template Entrance Channel as Possible Allosteric Inhibition and Resistance Site for Quinolines Tricyclic Derivatives in RNA Dependent RNA Polymerase of Bovine Viral Diarrhea Virus;Pharmaceuticals;2023-03-01
4. Fluorescence Anisotropy-Based Assay for Characterization of Ligand Binding Dynamics to GPCRs: The Case of Cy3B-Labeled Ligands Binding to MC4 Receptors in Budded Baculoviruses;Methods in Molecular Biology;2021
5. Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M2 Receptor;Journal of Medicinal Chemistry;2020-04-01
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3