Abstract
The synthesis is described
of octahydro-1H-2-pyrindine-5,7-dione (4) and its 6-diazo and 6-bromo derivatives.
These are analogues of GABA in which the carboxyl group is replaced by an enolic β-diketone. The compounds showed negligible or
very weak activity as GABA agonists with respect to inhibition of [3H] GABA
binding, uptake and transamination in rat brain
membranes.
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