Crucial Aspects for Maintaining rAAV Stability

Author:

Lengler Johannes1,Gavrila Miruna1,Brandis Janina2,Palavra Kristina1,Dieringer Felix1,Unterthurner Sabine1,Fuchsberger Felix1,Kraus Barbara1,Bort Juan A. Hernandez1

Affiliation:

1. Gene Therapy Process Development, Baxalta Innovations GmbH, a part of Takeda companies

2. Drug Product Development EU, Baxalta Innovations GmbH, a part of Takeda companies

Abstract

Abstract

Background The storage of rAAV vectors for gene therapy applications is critical for ensuring a constant product quality and defined amount of medication at the time of administration. Therefore, we determined the influence of different storage conditions on the physicochemical and biological properties of rAAV8 and rAAV9 preparations. Particular attention was paid to short-term storage, which plays a crucial role in both the manufacturing process and in clinical applications. Additionally, we addressed the question, of viability of rAAV8 and rAAV9 when subjected to very low-temperature storage conditions (< -65°C) or lyophilization. To determine the impact on rAAV vectors, various analyses were used, including the quantification of capsid and genome titers, as well as biopotency assessments, which are pivotal determinants in characterizing vector behavior and efficacy. Results Our data showed that freeze/thaw cycles hardly affected the functionality of rAAV9-aGAL vectors. In contrast, prolonged storage at room temperature for several days, resulted in a discernible decrease in biopotency despite consistent capsid and genome titers. When the storage temperature was further increased, the rAAV8-aGAL decay accelerated. For example, a short-term exposure of + 40°C and more, led to a reduction in the physical viral titer and to an even faster decline in efficacy determined by biopotency. However, the addition of sucrose and sorbitol to the rAAV9-aGAL and rAAV9-GAA preparations reduced the temperature sensitivity of rAAV and improved its stability. Furthermore, exposure of rAAV9-aGAL to highly acidic conditions (pH 2.5) dramatically reduced its biopotency by 70% or more. Most interestingly, a long-term storage of rAAV9-aGAL and rAAV8-FVIII vectors over 12 months and 36 months, respectively, demonstrated exceptional stability at storage temperatures below − 65°C. Also lyophilization conserved functionality for at least 10 months. Conclusions Our data showed how to maintain rAAV biopotency levels over the time without substantial loss. Storage at very low temperatures (< -65°C) preserved its effectiveness over years. Overall, pH and temperature conditions during the manufacturing process, storage and clinical application are worth considering. Consistency in the rAAV capsid titer determination did not necessarily indicate the preservation of biopotency. In conclusion, our approach determined several options for maximizing rAAV stability.

Publisher

Springer Science and Business Media LLC

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