P-gp Inhibition Potential in Cell-Based Models: Which “Calculation” Method is the Most Accurate?
Author:
Publisher
Springer Science and Business Media LLC
Subject
Pharmaceutical Science
Link
http://link.springer.com/content/pdf/10.1208/s12248-008-9068-x.pdf
Reference26 articles.
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4. C. Matheny, M. Lamb, K. Brouwer, and G. Pollak. Pharmacokinetic and pharmacodynamic implications of P-gp modulation. Pharmacotherapy. 21:778–796 (2001).
5. J. Polli, et al. Role of P-gp on CNS disposition of amprenavir, an HIV protease inhibitor. Pharm. Res. 16:1206–1212 (1999).
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