Ligand- and mutation-induced conformational selection in the CCR5 chemokine G protein-coupled receptor
Author:
Publisher
Proceedings of the National Academy of Sciences
Subject
Multidisciplinary
Reference28 articles.
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1. The chemokine receptor CCR5: multi-faceted hook for HIV-1;Retrovirology;2024-01-23
2. Investigating the Effect of GLU283 Protonation State on the Conformational Heterogeneity of CCR5 by Molecular Dynamics Simulations;2023-08-18
3. Insight into the Structure and Physicochemical Properties of Potent Chemokine Receptor 5 Inhibitors for the Discovery of Novel Alzheimer’s Disease Drugs;Central Nervous System Agents in Medicinal Chemistry;2023-08
4. Intermediate-state-trapped mutants pinpoint G protein-coupled receptor conformational allostery;Nature Communications;2023-03-10
5. Tracking receptor motions at the plasma membrane reveals distinct effects of ligands on CCR5 dynamics depending on its dimerization status;eLife;2022-07-22
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