Irreversible inhibition of estrogen receptor α signaling and the emergence of hormonal resistance in MCF7 breast cancer cells induced by DNA damage agents

Author:

Scherbakov Alexander1,Sorokin Danila1,Razuvaeva Valeria1,Shchegolev Yuri1,Andreeva Olga1,Salnikova Diana1,Fetisov Timur2,Vlasova Olga2,Kirsanov Kirill2,Gudkova Margarita1,Krasil'nikov Mikhail1

Affiliation:

1. Department of Experimental Tumor Biology, Institute of Carcinogenesis, N.N. Blokhin National Medical Research Center of Oncology, The Ministry of Health of Russia, Moscow 115522, Russian Federation

2. Department of Chemical Carcinogenesis, Institute of Carcinogenesis, N.N. Blokhin National Medical Research Center of Oncology, The Ministry of Health of Russia, Moscow 115522, Russian Federation

Publisher

Spandidos Publications

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4. Design, synthesis, and biological evaluation of BRD4 degraders;Ding;Bioorg Med Chem,2023

5. Discovery of small molecule mechanistic target of rapamycin inhibitors as anti-aging and anti-cancer therapeutics;Chrienova;Front Aging Neurosci,2022

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