Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3H-pyrazolo[3,4-d]pyrimidin-3-one-Reference-Cited by-同舟云学术

Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3H-pyrazolo[3,4-d]pyrimidin-3-one

Published:2016-02-01 Issue:1 Volume:22 Page:49-53
ISSN:2191-0197
Container-title:Heterocyclic Communications
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Author:

Ebrahimpour Zahra¹,Shiri Ali¹,Bakavoli Mehdi¹,Seyedi Seyed Mohammad¹,Bahreini Masoumeh²,Oroojalian Fatemeh³

Affiliation:

1. 1Faculty of Science, Department of Chemistry, Ferdowsi University of Mashhad, 91775-1436 Mashhad, Iran (Islamic Republic of)

2. 2Faculty of Science, Department of Biology, Ferdowsi University of Mashhad, Mashhad, Iran (Islamic Republic of)

3. 3Faculty of New Sciences and Technologies, Department of Life Science Engineering, University of Tehran, 14395-1561 Tehran, Iran (Islamic Republic of)

Abstract

AbstractSynthesis of new 1,2-dihydro-3H-pyrazolo[3,4-d] pyrimidin-3-ones4–6starting with ethyl 4-hydroxy-2-methylthio-pyrimidine-5-carboxylate (1) under classical heating and microwave-induced conditions is reported. The antibacterial activities of the synthesized compounds were evaluated using chloramphenicol and streptomycin as reference drugs.

Publisher

Walter de Gruyter GmbH

Subject

Organic Chemistry

Link

https://www.degruyter.com/document/doi/10.1515/hc-2015-0145/pdf

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