Process Development and Large-Scale Synthesis of NK1 Antagonist
Author:
Affiliation:
1. Research Center, Kyorin Pharmaceutical Co., Ltd.
2. Faculty of Pharmaceutical Sciences, Toho University
Publisher
Pharmaceutical Society of Japan
Subject
Drug Discovery,General Chemistry,General Medicine
Link
http://www.jstage.jst.go.jp/article/cpb/56/2/56_2_176/_pdf
Reference18 articles.
1. Tachykinin receptor types: Classification and membrane signalling mechanisms
2. An unidentified depressor substance in certain tissue extracts
3. The role of peptides in the regulation of the micturition reflex: An update
4. Evidence for a role of tachykinins as sensory transmitters in the activation of micturition reflex
5. Design, synthesis, and evaluation of novel 2-substituted-4-aryl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,5]oxazocin-5-ones as NK1 antagonists
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3. Efficient and Benign One-Pot Conversion of N-Tosyl-1,4,5,6-tetrahydropyrimidines to Pyrimidines via Tandem β-Elimination and Aromatization;Synthetic Communications;2013-09-04
4. ChemInform Abstract: Process Development and Large-Scale Synthesis of NK1Antagonist.;ChemInform;2008-08-05
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