The potency of selatogrel, a reversible antagonist of the P2Y12 receptor, is affected by calcium concentration
Author:
Affiliation:
1. Drug Discovery Biology, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland
Publisher
Informa UK Limited
Subject
Hematology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/09537104.2020.1869711
Reference47 articles.
1. Historical perspective and future directions in platelet research
2. Intramyocardial platelet aggregation in patients with unstable angina suffering sudden ischemic cardiac death.
3. The central role of the P 2T receptor in amplification of human platelet activation, aggregation, secretion and procoagulant activity
4. Updates and Current Recommendations for the Management of Patients With Non–ST-Elevation Acute Coronary Syndromes: What It Means for Clinical Practice
5. Management of Patients With NSTE-ACS
Cited by 8 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Clinical pharmacology of selatogrel for self-administration by patients with suspected acute myocardial infarction;Expert Opinion on Drug Metabolism & Toxicology;2023-10-03
2. Mind the Gap: Model-Based Switching from Selatogrel to Maintenance Therapy with Oral P2Y12 Receptor Antagonists;Biomolecules;2023-09-08
3. Recent advances in targeting the “undruggable” proteins: from drug discovery to clinical trials;Signal Transduction and Targeted Therapy;2023-09-06
4. Comparison of the effects of the GPIIb-IIIa antagonist Zalunfiban and the P2Y12 antagonist Selatogrel on Platelet Aggregation;Journal of Thrombosis and Thrombolysis;2023-08-10
5. Inverse agonist efficacy of selatogrel blunts constitutive P2Y12 receptor signaling by inducing the inactive receptor conformation;Biochemical Pharmacology;2022-12
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3