Ligand-based design and synthesis of N'-Benzylidene-3,4-dimethoxybenzohydrazide derivatives as potential antimicrobial agents; evaluation by in vitro, in vivo, and in silico approaches with SAR studies-Reference-Cited by-同舟云学术

Ligand-based design and synthesis of N'-Benzylidene-3,4-dimethoxybenzohydrazide derivatives as potential antimicrobial agents; evaluation by in vitro, in vivo, and in silico approaches with SAR studies

Published:2022-04-18 Issue:1 Volume:37 Page:1098-1119
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Ezz Eldin Rogy R.¹,Saleh Marwa A.²^ORCID,Alotaibi Mohammad Hayal³,Alsuair Reem K.³,Alzahrani Yahya A.³,Alshehri Feras A.³,Mohamed Amany F.⁴,Hafez Shaimaa M.⁴,Althoqapy Azza Ali⁵,Khirala Seham K.⁵,Amin Mona M.⁶,A. F Yousuf⁷,AbdElwahab Azza H.⁷,Alesawy Mohamed S.⁸,Elmaaty Ayman Abo⁹,Al-Karmalawy Ahmed A.¹⁰^ORCID

Affiliation:

1. Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Port Said University, Port Said, Egypt

2. Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo, Egypt

3. National Center for Chemical Technologies, King Abdulaziz City for Science and Technology, Riyadh, Saudi Arabia

4. Department of Anatomy and Embryology, Faculty of Medicine for Girls, Al-Azhar University, Cairo, Egypt

5. Department of Microbiology and Immunology, Faculty of Medicine for Girls, Al-Azhar University, Cairo, Egypt

6. Department of Pharmacology, Faculty of Medicine for Girls, Al-Azhar University, Cairo, Egypt

7. Department of Physiology, Faculty of Medicine for Girls, Al-Azhar University, Cairo, Egypt

8. Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Boys), Al‐Azhar University, Cairo, Egypt

9. Department of Medicinal Chemistry, Faculty of Pharmacy, Port Said University, Port Said, Egypt

10. Department of Pharmaceutical Medicinal Chemistry, Faculty of Pharmacy, Horus University-Egypt, New Damietta, Egypt

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2063282

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