Discovery of a new class of triazole based inhibitors of acetyl transferase KAT2A

Author:

Pacifico Roberta1,Del Gaudio Nunzio2,Bove Guglielmo2,Altucci Lucia2ORCID,Siragusa Lydia3,Cruciani Gabriele4,Ruvo Menotti5ORCID,Bellavita Rosa6ORCID,Grieco Paolo6ORCID,Adamo Mauro F. A.1ORCID

Affiliation:

1. Centre for Synthesis and Chemical Biology (CSCB), Department of Chemistry, Royal College of Surgeons in Ireland, Dublin, Ireland

2. Department of precision medicine, University of Campania Luigi Vanvitelli, Naples, Italy

3. Molecular Horizon Srl, Bettona, Italy

4. Laboratory for Chemometrics and Molecular Modeling, Department of Chemistry, Biology, and Biotechnology, University of Perugia, Perugia, Italy

5. Institute of Biostructures and Bioimaging, Consiglio Nazionale delle Ricerche, Naples, Italy

6. Department of Pharmacy, School of Medicine, University of Naples ‘Federico II’, Naples, Italy

Funder

Irish Research Council

VALERE

Programma Operativo Nazionale Ricerca e Competitività

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

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