Design, synthesis, and biological evaluation of triazole-pyrimidine-methylbenzonitrile derivatives as dual A2A/A2B adenosine receptor antagonists
Author:
Affiliation:
1. School of Pharmacy, Binzhou Medical University, Yantai, China
2. Luye Pharma Group, Yantai, China
Funder
Projects of Medical and Health Technology Development Program
the Scientific Research Foundation of Binzhou Medical University
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2077731
Reference41 articles.
1. Adenosine A2A Receptor Antagonists for Cancer Immunotherapy
2. Adenosine receptor antagonists: Recent advances and therapeutic perspective
3. Novel positive allosteric modulators of A2B adenosine receptor acting as bone mineralisation promoters
4. Design, synthesis and biological evaluation of novel scaffold benzo[4,5]imidazo [1,2-a]pyrazin-1-amine: Towards adenosine A2A receptor (A2A AR) antagonist
5. The aminopyridine-3,5-dicarbonitrile core for the design of new non-nucleoside-like agonists of the human adenosine A2B receptor
Cited by 6 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Structural modification strategies of triazoles in anticancer drug development;European Journal of Medicinal Chemistry;2024-09
2. A Review of Recent Progress on the Anticancer Activity of Heterocyclic Compounds;SynOpen;2024-08
3. Unlocking the adenosine receptor mechanism of the tumour immune microenvironment;Frontiers in Immunology;2024-06-27
4. PI3Kδ and mTOR dual inhibitors: Design, synthesis and anticancer evaluation of 3-substituted aminomethylquinoline analogues;Bioorganic Chemistry;2024-06
5. Adenosine A2A Receptor Antagonists: Chemistry, SARs, and Therapeutic Potential;Topics in Medicinal Chemistry;2023
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3