Discovery of 2,4-thiazolidinedione-tethered coumarins as novel selective inhibitors for carbonic anhydrase IX and XII isoforms

Author:

Eldehna Wagdy M.1,Taghour Mohammed S.2,Al-Warhi Tarfah3,Nocentini Alessio4ORCID,Elbadawi Mostafa M.1,Mahdy Hazem A.2,Abdelrahman Mohamed A.5,Alotaibi Ohoud J.3,Aljaeed Nada3,Elimam Diaaeldin M.67,Afarinkia Kamyar8,Abdel-Aziz Hatem A.9,Supuran Claudiu T.4ORCID

Affiliation:

1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt

2. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy, Al-Azhar University, Cairo, Egypt

3. Department of Chemistry, College of Science, Princess Nourah Bint Abdulrahman University, Riyadh, Saudi Arabia

4. Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy

5. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Egyptian Russian University, Cairo, Egypt

6. Department of Pharmacognosy, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt

7. School of Molecular and Cellular Biology, Faculty of Biological Sciences, University of Leeds, Leeds, United Kingdom

8. Institute of Cancer Therapeutics, University of Bradford, Bradford, United Kingdom

9. Department of Applied Organic Chemistry, National Research Center, Giza, Egypt

Funder

Deanship of Scientific Research at Princess Nourah bint Abdulrahman University

Italian Ministry for Education and Science

Ente Cassa di Risparmio di Firenze

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

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