Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity-Reference-Cited by-同舟云学术

Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivity

Published:2023-04-20 Issue:1 Volume:38 Page:
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Allam Heba Abdelrasheed¹,Albakry Mohamed E.²,Mahmoud Walaa R.¹,Bonardi Alessandro³,Moussa Shaimaa A.¹,Mohamady Samy⁴,Abdel-Aziz Hatem A.⁵,Supuran Claudiu T.³^ORCID,Ibrahim Hany S.²⁶^ORCID

Affiliation:

1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Giza, Egypt

2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Egyptian Russian University, Badr City, Egypt

3. Department of NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Florence, Italy

4. Faculty of Pharmacy, The British University in Egypt, El Shorouk, Egypt

5. Department of Applied Organic Chemistry, National Research Center, Giza, Egypt

6. Department of Medicinal Chemistry, Institute of Pharmacy, Martin-Luther-University of Halle-Wittenberg, Halle (Saale), Germany

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2023.2201403

Reference44 articles.

1. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

2. The γ class of carbonic anhydrases

3. Thylakoid luminal θ-carbonic anhydrase critical for growth and photosynthesis in the marine diatom Phaeodactylum tricornutum

4. Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases

5. Structural and inhibition insights into carbonic anhydrase CDCA1 from the marine diatom Thalassiosira weissflogii

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