Energetically optimized pharmacophore modeling to identify dual negative allosteric modulators against group I mGluRs in neurodegenerative diseases
Author:
Affiliation:
1. Computer Aided Drug Designing and Molecular Modeling Laboratory, Department of Bioinformatics, Alagappa University, Karaikudi, India
Publisher
Informa UK Limited
Subject
Molecular Biology,General Medicine,Structural Biology
Link
https://www.tandfonline.com/doi/pdf/10.1080/07391102.2019.1640794
Reference41 articles.
1. Pharmacophore and structure-based drug design, molecular dynamics and admet/tox studies to design novel potential pad4 inhibitors
2. Opportunities and Challenges in the Discovery of Allosteric Modulators of GPCRs
3. Group I metabotropic glutamate receptors activate a calcium‐sensitive transient receptor potential‐like conductance in rat hippocampus
4. Differential distribution of group I metabotropic glutamate receptors in developing human cortex
5. Drug Design Strategies for GPCR Allosteric Modulators
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