Design, Synthesis and In Vitro Evaluation of Novel Benzo[b]thiophene Derivatives as Serotonin N-acetyltransferase (AANAT) Inhibitors
Author:
Affiliation:
1. Laboratoire de Chimie Thérapeutique, Faculté des Sciences Pharmaceutiques et Biologiques, BP 83 59006, Lille Cedex, France
2. Institut de Recherches Internationales Servier, 6 place des pléiades, 92415, Courbevoie Cedex, France
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/1475636031000093552
Reference11 articles.
1. Melatonin, Its Receptors, and Relationships with Biological Rhythm Disorders
2. Melatonin and sleep in humans
3. Kinetic Analysis of the Catalytic Mechanism of Serotonin N-Acetyltransferase (EC 2.3.1.87)
4. A Potent Inhibitor of the Melatonin Rhythm Enzyme
Cited by 11 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. How Can Molecular Pharmacology Help Understand the Multiple Actions of Melatonin: 20 Years of Research and Trends;Melatonin - Molecular Biology, Clinical and Pharmaceutical Approaches;2018-11-21
2. Theoretical evaluation and improvement on the potency of the rhodanine-based inhibitors for human serotoninN-acetyltransferase;Molecular Simulation;2014-01-16
3. Electrosynthesis of Fluorinated Benzo[b]thiophene Derivatives;Synlett;2011-05-05
4. Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands;European Journal of Medicinal Chemistry;2011-05
5. Utility of 3-Chlorobenzothiophene-2-Carbonylisothiocyanate for the Synthesis of Some Novel Biheterocycles of Expected Biological Activity;Phosphorus, Sulfur, and Silicon and the Related Elements;2010-06-30
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3