Chemical synthesis and in vitro biological evaluation of a phosphorylated bisubstrate inhibitor of type 3 17β-hydroxysteroid dehydrogenase
Author:
Affiliation:
1. Medicinal Chemistry Division, Oncology and Molecular Endocrinology Research Center, CHUQ-Pavillon CHUL and Université Laval, Québec, G1V 4G2, Canada
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/14756360601051423
Reference33 articles.
1. Analysis and characteristics of multiple types of human 17β-hydroxysteroid dehydrogenase
2. Intracrinology: role of the family of 17 beta-hydroxysteroid dehydrogenases in human physiology and disease
3. Role of 17β-Hydroxysteroid Dehydrogenases in Sex Steroid Formation in Peripheral Intracrine Tissues
4. The role of 17 beta-hydroxysteroid dehydrogenases
5. Male pseudohermaphroditism caused by mutations of testicular 17β–hydroxysteroid dehydrogenase 3
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