Efficient library synthesis of imidazoles using a multicomponent reaction and microwave irradiation
-
Published:2006-02
Issue:1
Volume:10
Page:17-22
-
ISSN:1381-1991
-
Container-title:Molecular Diversity
-
language:en
-
Short-container-title:Mol Divers
Author:
Gelens E.,Kanter F. J. J. De,Schmitz R. F.,Sliedregt L. A. J. M.,Steen B. J. Van,Kruse Chris G.,Leurs R.,Groen M. B.,Orru R. V. A.
Publisher
Springer Science and Business Media LLC
Subject
Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Drug Discovery,Molecular Biology,General Medicine,Information Systems,Catalysis
Reference25 articles.
1. Kitbunnadaj, R., Zuiderveld, O.P., Christophe, B., Hulscher, S., Menge, W.M.P.B., Gelens, E., Snip, E., Bakker, R.A., Celanire, S., Gillard, M., Talaga, P., Timmerman, H. and Leurs, R., Identification of 4-(1H-imidazol-4(5)-ylmethyl)pyridine (immethridine) as a novel, potent, and highly selective histamine H-3 receptor agonist, J. Med. Chem., 10 (2004) 2414–2417. 2. Adams, J.L., Boehm, J.C., Gallagher, T.F., Kassis, S., Webb, E.F., Hall, R., Sorenson, M., Garigipati, R., Griswold, D.E. and Lee, J.C., Pyrimidinylimidazole inhibitors of p38: Cyclic N-1 imidazole substituents enhance p38 kinase inhibition and oral activity, Bioog. Med. Chem. Lett., 11 (2001) 2867–2870. 3. Dinsmore, C.J., Williams, T.M., O'Neill, A.B., Liu, D., Rands, E., Culberson, J.C., Lobell, R.B., Koblan, K.S., Kohl, N.E., Gibbs, J.B., Oliff, A.I., Graham, S.L. and Hartman, G.D., Imidazole-containing diarylether and diarylsulfone inhibitors of farnesyl-protein transferase Bioog. Med. Chem. Lett., 9 (1999) 3301–3306. 4. Khanna, I.K., Weier, R.M., Yu, Y., Xu, X.D., Kosyk, F.J., Collins, P.W., Koboldt, C.M., Veenhuizen, A.W., Perkins, W.E., Casler, J.J., Masferrer, J.L., Zhang, Y.Y., Gregory, S.A., Seibert, K. and Isakson, P.C., 1,2-Diarylimidazoles as potent, cycloogygenase-2 selective, and orally active antiinflammatory agents, J. Med. Chem., 40 (1997) 1634–1647. 5. Revesz, L., Bonne, F. and Makavou, P., Vicinal bromostannanes as novel building blocks for the preparation of di- and trisubstituted imidazoles, Tetrahedron Lett., 39 (1998) 5171–5174.
Cited by
69 articles.
订阅此论文施引文献
订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Synthesis and Reactions of 3‐Amino‐5,6‐Dimethyl‐l,2,4‐Triazine: DFT Studies, ADME Assay, and Molecular Docking on the new l,2,4‐Triazine Derivatives as Anticancer Agents.;ChemistrySelect;2024-04-22 2. Synthesis of Heterocyclic Compounds Under Microwave Irradiation Using Name Reactions;Green Chemical Synthesis with Microwaves and Ultrasound;2024-03-28 3. Vitamin C as an Effective Organocatalyst for Three and Four‐Component Synthesis of 1,2,4,5‐tetrasubstituted Imidazoles;ChemistrySelect;2023-10-02 4. Design, synthesis of novel substituted imidazole derivatives: Cytotoxicity and molecular docking studies;Chemical Data Collections;2023-10 5. Brønsted Acid-Catalyzed Synthesis of 1,2,5-Trisubstituted Imidazoles via a Multicomponent Reaction of Vinyl Azides with Aromatic Aldehydes and Aromatic Amines;The Journal of Organic Chemistry;2022-10-12
|
|