PK/PD studies on non-selective PDE inhibitors in rats using cAMP as a marker of pharmacological response
Author:
Funder
Uniwersytet Jagielloński Collegium Medicum
Publisher
Springer Science and Business Media LLC
Subject
Pharmacology,General Medicine
Link
http://link.springer.com/article/10.1007/s00210-017-1406-z/fulltext.html
Reference65 articles.
1. Amado J, Fidalgo I, García-Unzueta M et al (1999) Patients with poor preoperative ejection fraction have a higher plasma response of adrenomedullin in response to open heart surgery. Acta Anaesthesiol Scand 43:829–833. doi: 10.1034/j.1399-6576.1999.430808.x
2. Ariens EJ, Van Rossum JM, Simonis AM (1957) Affinity, intrinsic activity and drug interactions. Pharmacol Rev 9:218–236
3. Bai JPF, Bell R, Buckman S et al (2011) Translational biomarkers: from preclinical to clinical a report of 2009 AAPS/ACCP biomarker workshop. AAPS J 13:274–283. doi: 10.1208/s12248-011-9265-x
4. Bian H, Zhang J, Wu P et al (2004) Differential type 4 cAMP-specific phosphodiesterase (PDE4) expression and functional sensitivity to PDE4 inhibitors among rats, monkeys and humans. Biochem Pharmacol 68:2229–2236. doi: 10.1016/j.bcp.2004.08.014
5. Bleich D, Chen S, Bursten SL, Nadler JL (1996) Lisofylline, an inhibitor of unsaturated phosphatidic acid generation, ameliorates interleukin-1 beta-induced dysfunction in cultured rat islets. Endocrinology 137:4871–4877. doi: 10.1210/endo.137.11.8895359
Cited by 14 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Therapeutic perspectives on PDE4B inhibition in adipose tissue dysfunction and chronic liver injury;Expert Opinion on Therapeutic Targets;2024-06-19
2. The effect of a methylxanthine vasodilator: pentoxifylline on the treatment of diabetic nephropathy—a meta-analysis;Naunyn-Schmiedeberg's Archives of Pharmacology;2023-11-21
3. Pharmacokinetic/Pharmacodynamic Assessment of Selective Phosphodiesterase Inhibitors in a Mouse Model of Autoimmune Hepatitis;Journal of Pharmacology and Experimental Therapeutics;2022-02-27
4. Chemoenzymatic deracemization of lisofylline catalyzed by a (laccase/TEMPO)-alcohol dehydrogenase system;Catalysis Science & Technology;2022
5. PK/PD Modeling of the PDE7 Inhibitor—GRMS-55 in a Mouse Model of Autoimmune Hepatitis;Pharmaceutics;2021-04-21
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3