Phase II trial of multi-kinase inhibitor ESK981 in patients with metastatic castration-resistant prostate cancer
Author:
Publisher
Springer Science and Business Media LLC
Link
https://link.springer.com/content/pdf/10.1007/s10637-024-01463-x.pdf
Reference20 articles.
1. Ferraldeschi R, Pezaro C, Karavasilis V, de Bono J (2013) Abiraterone and novel antiandrogens: overcoming castration resistance in prostate cancer. Annu Rev Med 64:1–13. https://doi.org/10.1146/annurev-med-121211-091605
2. Ryan CJ, Smith MR, de Bono JS, Molina A, Logothetis CJ, de Souza P et al (2013) Abiraterone in metastatic prostate cancer without previous chemotherapy. N Engl J Med 368:138–148. https://doi.org/10.1056/NEJMoa1209096
3. Scher HI, Fizazi K, Saad F, Taplin ME, Sternberg CN, Miller K et al (2012) Increased survival with enzalutamide in prostate cancer after chemotherapy. N Engl J Med 367:1187–1197. https://doi.org/10.1056/NEJMoa1207506
4. Qiao Y, Choi JE, Tien JC, Simko SA, Rajendiran T, Vo JN et al (2021) Autophagy Inhibition by Targeting PIKfyve Potentiates Response to Immune Checkpoint Blockade in Prostate Cancer. Nat Cancer 2:978–993. https://doi.org/10.1038/s43018-021-00237-1
5. Pili R, Carducci M, Brown P, Hurwitz H (2014) An open-label study to determine the maximum tolerated dose of the multitargeted tyrosine kinase inhibitor CEP-11981 in patients with advanced cancer. Invest New Drugs 32:1258–1268. https://doi.org/10.1007/s10637-014-0147-9
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