Improvement of Oral Bioavailability of N-251, a Novel Antimalarial Drug, by Increasing Lymphatic Transport with Long-Chain Fatty Acid-Based Self-Nanoemulsifying Drug Delivery System

Author:

Imada Chikako,Takahashi Takuma,Kuramoto Makoto,Masuda Kazufumi,Ogawara Ken-ichi,Sato Akira,Wataya Yusuke,Kim Hye-Sook,Higaki Kazutaka

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Organic Chemistry,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biotechnology

Reference38 articles.

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2. Fujioka Y, Kadono K, Fujie Y, Metsugi Y, Ogawara K, Higaki K, et al. Prediction of oral absorption of griseofulvin, a BCS class II drug, based on GITA model: utilization of a more suitable medium for in-vitro dissolution study. J Control Rel. 2008;352:36–43.

3. Fujioka Y, Metsugi Y, Ogawara K, Higaki K, Kimura T. Evaluation of in-vivo dissolution behavior and GI transit of griseofulvin, a BCS class II drug. Int J Pharm. 2008;352:36–43.

4. Serajuddin ATM. Solid dispersion of poorly water-soluble drugs: early promises, subsequent problems, and recent breakthroughs. J Pharm Sci. 1999;88:1058–66.

5. Grove M, Müllertz A. Liquid self-microemulsifying drug delivery system. In: Hauss DJ, editor. Oral lipid-based formulations. New York: Informa; 2007. p. 107–27.

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