QSAR analysis of centrally fused 1,5-diaryl pyrazoles for cyclooxygenase inhibition using MOE-Qua-SAR descriptors
Author:
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
http://link.springer.com/content/pdf/10.1007/s00044-008-9136-x.pdf
Reference19 articles.
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2. Botting JH (1999) Nonsteroidal antiinflammatory agents. Drugs Today (Barc) 35:225–235
3. Dannhardt G, Kiefer W (2000) Cyclooxygenase inhibitors—current status and future prospectus. Eur J Med Chem 36:109–126. doi: 10.1016/S0223-5234(01)01197-7
4. Garg R, Kurup A, Mekapati SB, Hansch C (2003) Cycloxygenase (COX) inhibitors: a comparative QSAR study. Chem Rev 103:703–731. doi: 10.1021/cr020464a
5. Kurumbail RG, Pak JY, Gildehaus D, Miyashiro JM, Stevens AM, Gierse JK et al (1996) Structural basis for selective inhibition of cyclooxygenase-2 by antiinflammatory agents. Nature 384:644–648. doi: 10.1038/384644a0
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