Current trends and future directions for the synthesis and pharmacological applications of 2-(2-cyanopyrrolidin-1-yl)-N-3-hydroxyadamantan-1-yl) acetamide (Gliptins)
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Publisher
Springer Science and Business Media LLC
Link
https://link.springer.com/content/pdf/10.1007/s00044-024-03218-y.pdf
Reference41 articles.
1. Lai ZW, Li C, Liu J, Kong L, Wen X, Sun H. Discovery of highly potent DPP-4 inhibitors by hybrid compound design based on linagliptin and alogliptin. Eur J Med Chem. 2014;83:547–60. https://doi.org/10.1016/j.ejmech.2014.06.044
2. Sneha P, Doss CGP. Gliptins in managing diabetes - reviewing computational strategy. Life Sci. 2016;166:108–20. https://doi.org/10.1016/j.lfs.2016.10.009
3. Hu N, Zhao G, Zhang Y, Liu X, Li G, Tang W. Synthesis of chiral α-amino tertiary boronic esters by enantioselective hydroboration of α-arylenamides. J Am Chem Soc. 2015;137:6746–9. https://doi.org/10.1021/jacs.5b03760
4. Plescia J, Moitessier N. Design and discovery of boronic acid drugs. Eur J Med Chem. 2020;195:112270. https://doi.org/10.1016/j.ejmech.2020.112270
5. Kim MK, Chae YN, Kim HD, Yang EK, Cho EJ, Choi SH, et al. DA-1229, a novel and potent DPP-4 inhibitor, improves insulin resistance and delays the onset of diabetes. Life Sci. 2012;90:21–29. https://doi.org/10.1016/j.lfs.2011.10.007
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