‘Polymorphism-aided’ Selective Targeting and Inhibition of Caspase-6 by a Novel Allosteric Inhibitor Towards Efficient Alzheimer’s Disease Treatment

Author:

Kumi Ransford Oduro,Agoni Clement,Issahaku Abdul Rashid,Olotu Fisayo A.,Soliman Mahmoud E. S.ORCID

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Biochemistry,General Medicine,Biophysics

Reference42 articles.

1. Deepak, K. (2018). Identification of FDA-approved drugs as novel allosteric inhibitors of human executioner caspases. Proteins, 86(11), 1202–1210.

2. Behzadi, P. (2015). Caspases and apoptosis. iMedPub Journal, 1(2), 6.

3. MacKenzie, S. H., Schipper, J. L., & Clark, A. C. (2010). The potential for caspases in drug discovery. Current Opinion in Drug Discovery and Development, 13(5), 568–576.

4. Howley, B., & Fearnhead, H. O. (2008). Caspases as therapeutic targets. Journal of Cellular and Molecular Medicine, 12(5A), 1502–1516.

5. Garrido, E. R., Heidt, L., Beaubier, N., & Troy, C. M. (2011). Neurochemical mechanisms in disease. Advances in Neurobiology 1, Springer New York, chapter 2, 17–47.

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