Refining Efficacy: Allosterism and Bias in G Protein-Coupled Receptor Signaling
Author:
Publisher
Humana Press
Link
http://link.springer.com/content/pdf/10.1007/978-1-61779-160-4_1
Reference154 articles.
1. Stephenson, R. P. (1956) A modification of receptor theory. Br J Pharmacol 11, 379–93.
2. Black, J. W., and Leff, P. (1983) Operational models of pharmacological agonist. Proc R Soc Lond [Biol] 220, 141–62.
3. Black, J. W., Leff, P., and Shankley, N.P. (1985) An operational model of pharmacological agonism: The effect of E/[A] curve shape on agonist dissociation constant estimation. Br J Pharmacol 84, 561–71.
4. Kenakin, T., and Miller, L. E. (2010) Seven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery. Pharmacol Rev. 62, 265–304.
5. Koshland, D. E., Jr. (1998) Conformational changes: How small is big enough? Nature Med 4, 1112–4.
Cited by 73 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Probing phosphorylation events in biological membranes: The transducer function;Biochimica et Biophysica Acta (BBA) - Biomembranes;2024-10
2. Structural vulnerability in EPCR suggests functional modulation;Scientific Reports;2024-01-31
3. Arrestin and G Protein Interactions with GPCRs: A Structural Perspective;GPCRs as Therapeutic Targets;2022-09-16
4. Gene and protein interaction network analysis in the epithelial-mesenchymal transition of Hertwig's Epithelial Root Sheath reveals periodontal regenerative drug targets – An in silico study;Saudi Journal of Biological Sciences;2022-05
5. Structure of EPCR in a non-canonical conformation;2021-12-17
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3