Advances in Studies on Collagenase Inhibitors
Author:
Publisher
Springer Basel
Link
http://link.springer.com/content/pdf/10.1007/978-3-0348-0364-9_4.pdf
Reference108 articles.
1. Almstead NG, Bradley RS, Pikul S, De B, Natchus MG, Taiwo YO, Gu F, Williams LE, Hynd BA, Janusz MJ, Dunaway MC, Mieling GE (1999) Design, synthesis, and biological evaluation of potent thiazine and thiazepine based matrix metalloproteinase inhibitors. J Med Chem 42:4547–4562. doi: 10.1021/jm990330y
2. Aschia M, Roccatanoa D, Nolab AD, Gallinac C, Gavuzzod E, Pochettid G, Piepere M, Tscheschee H, Mazzaa F (2002) Computational study of the catalytic domain of human neutrophil collagenase. Specific role of the S3 and S’3 subsites in the interaction with a phosphonate inhibitor. J Comput Aided Mol Des 16:213–225
3. Baxter AD, Bhogal R, Bird J, Keily JF, Manallack DT, Montana JG, Owen DA, Pitt WR, Watson RJ, Wills RE (2001) Arylsulphonyl hydroxamic acids: potent and selective matrix metalloproteinase inhibitors. Bioorg Med Chem Lett 11:1465–1468
4. Becker DP, Barta TE, Bedell L, DeCrescenzo G, Freskos J, Getman DP, Hockerman SL, Li M, Mehta P, Mischke B, Munie GE, Swearingen C, Villamil CI (2001) alpha-Amino-beta-sulphone hydroxamates as potent MMP-13 inhibitors that spare MMP-1. Bioorg Med Chem Lett 11:2719–2722
5. Bertini I, Calderone V, Fragai M, Luchinat C, Mangani S, Terni B (2003) X-ray structures of binary and ternary enzyme-product-inhibitor complexes of matrix metalloproteinases. Angew Chem Int Ed Engl 42:2673–2676
Cited by 5 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Recent developments and strategies for the discovery of TACE inhibitors;Expert Opinion on Drug Discovery;2020-04-13
2. Design of selective TACE inhibitors using molecular docking studies: Synthesis and preliminary evaluation of anti-inflammatory and TACE inhibitory activity;SAR and QSAR in Environmental Research;2015-11-02
3. SAR Studies of Exosite-Binding Substrate-Selective Inhibitors of A Disintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes;Journal of Medicinal Chemistry;2015-08-04
4. QSAR Studies on Hydroxamic Acids: A Fascinating Family of Chemicals with a Wide Spectrum of Activities;Chemical Reviews;2015-05-29
5. Targeting of ECM molecules and their metabolizing enzymes and receptors for the treatment of CNS diseases;Progress in Brain Research;2014
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3